SULFA.org Independent · Reference

List of sulfa drugs.

A sulfa drug is any medication carrying the sulfonamide group –SO2NH2. Dozens of drugs qualify, but they do not all matter equally to someone with a sulfa allergy. The list below is split by the feature that actually predicts cross-reaction: whether the molecule also carries an arylamine at the N4 position. Sulfa antibiotics do. Almost nothing else does.

Educational reference — not medical advice. This page describes what is generally known about a drug family. It cannot account for your history, your other medicines, or your circumstances. Decisions about your own treatment belong with your doctor or pharmacist.

The short answer
If someone says "sulfa drug" without qualification, they mean a sulfa antibiotic — most often sulfamethoxazole/trimethoprim (Bactrim, Septra).
The dividing line
The N4 arylamine. Present in sulfa antibiotics and sulfasalazine; absent in the diuretics, sulfonylureas, celecoxib, and the carbonic anhydrase inhibitors.
Why it matters
An allergy label earned from a sulfa antibiotic does not automatically rule out the drugs in the second table. Cross-reactivity is low.

Group 1: sulfa antibiotics (arylamine-bearing)

These are the drugs that carry essentially the whole allergy burden. They carry the N4 arylamine, which the body oxidises to a reactive nitroso metabolite that binds to host proteins and provokes a drug-specific T-cell response. That pathway is well characterised, and it is the part of the structural argument that the evidence actually supports. (These drugs also share an N1 heterocyclic ring, sometimes proposed as the target of IgE-mediated reactions, but that is a hypothesis rather than a demonstrated mechanism.)

Antibiotic sulfonamides and close relatives
DrugCommon brandsUsed for
Sulfamethoxazole / trimethoprimBactrim, Septra, co-trimoxazoleUTI, MRSA skin infection, PCP prophylaxis, travellers' diarrhoea
SulfadiazineToxoplasmosis (with pyrimethamine), rheumatic fever prophylaxis
Silver sulfadiazine (topical)Silvadene, FlamazineBurn wound care
Sulfacetamide (topical / eye)Bleph-10, KlaronBacterial conjunctivitis, acne, seborrhoeic dermatitis
Sulfadoxine / pyrimethamineFansidarMalaria (limited, region-specific use)
SulfisoxazoleGantrisinLargely withdrawn; historical UTI agent
SulfasalazineAzulfidine, SalazopyrinUlcerative colitis, rheumatoid arthritis — not an antibiotic, but metabolised to arylamine-bearing sulfapyridine
Sulfasalazine is the exception worth remembering. It is prescribed as an anti-inflammatory, not an antibiotic, so it is easy to file mentally with the "safe" non-antibiotic sulfonamides. Chemically it does not belong there: the gut splits it into 5-ASA and sulfapyridine, and sulfapyridine carries the same arylamine as the antibiotics. People with a genuine sulfa antibiotic allergy may react to it. More on sulfasalazine.

Group 2: non-antibiotic sulfonamides (no arylamine)

Every drug below contains a sulfonamide group, which is why drug-interaction checkers and older references flag them against a "sulfa allergy." None of them carries the N4 arylamine. Published cross-reactivity rates are low, and most prescribers will use these drugs in a patient whose sulfa allergy came from a typical antibiotic rash.

Non-antibiotic sulfonamides by class
ClassDrugsUsed for
Loop diureticsFurosemide (Lasix), bumetanide, torsemideHeart failure, oedema
Thiazide & thiazide-like diureticsHydrochlorothiazide, chlorthalidone, indapamide, metolazone, chlorothiazideHigh blood pressure, oedema
SulfonylureasGlipizide, glyburide (glibenclamide), glimepiride, gliclazide, chlorpropamide, tolbutamideType 2 diabetes
Carbonic anhydrase inhibitorsAcetazolamide (Diamox), methazolamide, dorzolamide, brinzolamideGlaucoma, idiopathic intracranial hypertension, altitude sickness
COX-2 inhibitorCelecoxib (Celebrex)Arthritis, pain
TriptansSumatriptan, naratriptanMigraine
AnticonvulsantZonisamideEpilepsy
AntiarrhythmicsSotalol, dofetilide, ibutilideAtrial fibrillation and other arrhythmias
Alpha-blockerTamsulosinBenign prostatic hyperplasia
Endothelin antagonistsBosentan, macitentanPulmonary arterial hypertension
HIV protease inhibitorsDarunavir, fosamprenavir, tipranavirHIV treatment
UricosuricProbenecidGout
How prescribers generally treat this list. A patient whose record says "sulfa allergy" from a rash on Bactrim years ago is, in most modern practice, offered furosemide, HCTZ, glipizide, acetazolamide, or celecoxib without special ceremony. A patient whose past reaction was anaphylaxis, Stevens-Johnson syndrome, or DRESS is handled individually and cautiously. The severity of the original reaction, not the presence of a sulfonamide group, is what drives the decision. Mild versus severe reactions.

Frequently mistaken for sulfa drugs

Several drugs and substances end up on informal "avoid with sulfa allergy" lists without belonging there.

Not sulfonamides
SubstanceWhat it actually is
DapsoneA sulfone, not a sulfonamide — a different chemical class. The 2022 AAAAI/ACAAI practice parameter groups it with the drugs of minimal cross-reactivity concern after a sulfa antibiotic reaction. Its bigger issue is haemolysis in G6PD deficiency, which is why pre-prescription testing is standard.
TopiramateA sulfamate ester. Related but structurally distinct from a sulfonamide.
SulfitesFood and drug preservatives (wine, dried fruit, some injectables). Chemically unrelated to sulfa drugs.
SulfatesInorganic salts — magnesium sulfate, ferrous sulfate, sodium lauryl sulfate. Unrelated.
Elemental sulfurThe element, including sulfur-containing amino acids in food and sulfur in acne preparations. Unrelated.
Penicillins and cephalosporinsBeta-lactams. They contain a sulfur atom in the ring, which is not the same as a sulfonamide group. A sulfa allergy does not imply a penicillin allergy.

The overlap in names does real damage. Patients decline wine, avoid magnesium supplements, or refuse an antibiotic they could safely take, all on the strength of three shared letters. The disambiguation page works through each one.

How to use this list

The list identifies what contains a sulfonamide group. It does not tell you what is safe for you — that depends on what your original reaction actually was, how severe it was, and what alternatives exist for the condition being treated. If your record says "sulfa allergy" and you do not know the drug, the year, or the reaction, that is worth resolving: it is the single detail that determines how much of this list is genuinely off-limits. How to describe your allergy usefully, and how mislabelled allergies get removed.

References

  1. Khan DA, Banerji A, Blumenthal KG, et al. Drug allergy: a 2022 practice parameter update — Table XIV, drugs with no or weak evidence of cross-reactivity. J Allergy Clin Immunol. 2022;150(6):1333-93. www.jacionline.org
  2. Giles A, Foushee J, Lantz E, Gumina G. Sulfonamide allergies. Pharmacy (Basel). 2019;7(3):132. pmc.ncbi.nlm.nih.gov